Tibolone

Tibolone

Tibolone

Systematic (IUPAC) name

17-Hydroxy-7α-methyl-19-nor-17α-pregn-5(10)-en-20-yn-3-one

Identifiers

CAS number 5630-53-5

ATC code G03CX01

PubChem 21844

Chemical data

Formula C₂₁H₂₈O₂

Mol. mass 312.446 g/mol

Pharmacokinetic data

Bioavailability ?

Metabolism ?

Half life ?

Excretion ?

Therapeutic considerations

Pregnancy cat.
?

Legal status

Routes ?

Tibolone is a synthetic hormone-type drug. It is used mainly for hormone replacement therapy in post-menopausal women.

v • d • e

Sex hormones and related agents (primarily G03, also L02, H01C) – human endogenous in small caps

Agonist	PROGESTERONE · Dienogest · Desogestrel · Drospirenone · Dydrogesterone · Ethisterone · Etonogestrel · Ethynodiol diacetate · Gestodene · Gestonorone · Levonorgestrel · Lynestrenol · Medroxyprogesterone · Megestrol · Norelgestromin · Norethisterone · Norethynodrel · Norgestimate · Norgestrel · Norgestrienone · Tibolone

SPRM	Asoprisnil · CDB-4124

Antiprogestogen	Mifepristone

Agonist	TESTOSTERONE · Androstanolone · Fluoxymesterone · Mesterolone · Methyltestosterone · see also Anabolic steroids

Antiandrogen	Bicalutamide · Cyproterone · Dienogest · Flutamide · Nilutamide · Spironolactone

Agonist	ESTRADIOL · ESTRIOL · ESTRONE · Chlorotrianisene · Dienestrol · Diethylstilbestrol · Ethinylestradiol · Fosfestrol · Mestranol · Polyestradiol phosphate

SERM	Afimoxifene · Arzoxifene · Bazedoxifene · Clomifene · Fulvestrant · Lasofoxifene · Raloxifene · Tamoxifen · Toremifene

AI	Aminoglutethimide · Anastrozole · Atamestane · Exemestane · Fadrozole · Formestane · Letrozole · Vorozole

Antiestrogen	Mepitiostane

Agonist	Buserelin · Goserelin · Histrelin · Leuprorelin · Nafarelin · Triptorelin

Antagonist	Abarelix · Cetrorelix · Ganirelix

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